Accès direct Unités de recherche

Publications

Afficher tous

2014

Blond A, Ennifar E, Tisné C, Micouin L

The Design of RNA Binders: Targeting the HIV Replication Cycle as a Case Study. Article de journal

Dans: ChemMedChem, vol. 9, no. 9, p. 1982-96, 2014, ISBN: 25100137.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, RNA recognition antiviral agents drug design human immunodeficiency virus new targets, Unité ARN

Košutić M, Jud L, Veiga C Da, Frener M, Fauster K, Kreutz C, Ennifar E, Micura R

Surprising base pairing and structural properties of 2'-trifluoromethylthio-modified ribonucleic acids. Article de journal

Dans: J Am Chem Soc, vol. 136, no. 18, p. 6656-63, 2014, ISBN: 24766131.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

2013

Bec G, Meyer B, Gerard M A, Steger J, Fauster K, Wolff P, Burnouf D, Micura R, Dumas P, Ennifar E

Thermodynamics of HIV-1 Reverse Transcriptase in action elucidates the mechanism of action of non-nucleoside inhibitors. Article de journal

Dans: J Am Chem Soc, vol. 135, no. 26, p. 9743-9752, 2013, ISBN: 23742167.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Ennifar E

X-ray crystallography as a tool for mechanism-of-action studies and drug discovery Article de journal

Dans: Curr Pharm Biotechnol, vol. 14, no. 5, p. 537-550, 2013, ISBN: ISBN/1389-2010 (Print) 1873-4316 (Online).

Résumé | Liens | BibTeX | Étiquettes: Drug design Ligand Molecular mechanism Protein RNA Structural biology X-ray crystallography, DUMAS, ENNIFAR, Unité ARN

Ennifar E, Aslam M W, Strasser P, Hoffmann G, Dumas P, van Delft F L

Structure-guided Discovery of a Novel Aminoglycoside Conjugate Targeting HIV-1 RNA Viral Genome. Article de journal

Dans: ACS Chem Biol, vol. 8, no. 11, p. 2509-17, 2013, ISBN: 24015986.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Pendem N, Nelli Y R, Douat C, Fischer L, Laguerre M, Ennifar E, Kauffmann B, Guichard G

Controlling Helix Formation in the γ-Peptide Superfamily: Heterogeneous Foldamers with Urea/Amide and Urea/Carbamate Backbones Article de journal

Dans: Angew Chem Int Ed Engl, vol. 52, no. 15, p. 4147-51, 2013, ISBN: 23460200.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

2011

Heppell B, Blouin S, Dussault A M, Mulhbacher J, Ennifar E, Penedo J C, Lafontaine D A

Molecular insights into the ligand-controlled organization of the SAM-I riboswitch Article de journal

Dans: Nat Chem Biol, vol. 7, no. 6, p. 384-92, 2011, ISBN: ISBN/1552-4469 (Electronic) 1552-4450 (Linking), (Published online 01 May 2011).

Résumé | Liens | BibTeX | Étiquettes: Aptamers, Bacterial/*chemistry *Riboswitch S-Adenosylmethionine/*chemistry, DUMAS, ENNIFAR, Nucleotide/chemistry Bacillus subtilis/genetics Binding Sites Crystallography, Unité ARN, X-Ray Ligands Metals Nucleic Acid Conformation RNA

2010

Baussanne I, Bussiere A, Halder S, Ganem-Elbaz C, Ouberai M, Riou M, Paris J M, Ennifar E, Mingeot-Leclercq M P, Decout J L

Synthesis and antimicrobial evaluation of amphiphilic neamine derivatives Article de journal

Dans: J Med Chem, vol. 53, no. 1, p. 119-27, 2010, ISBN: 20000576, (1520-4804 (Electronic) 0022-2623 (Linking) Journal Article Research Support, Non-U.S. Gov't).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Ennifar E, Walter P, Dumas P

Cation-dependent cleavage of the duplex form of the subtype-B HIV-1 RNA dimerization initiation site Article de journal

Dans: Nucleic Acids Res, vol. 38, no. 17, p. 5807-5811, 2010, ISBN: 20460458, (1362-4962 (Electronic) 0305-1048 (Linking) Journal article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Fischer L, Claudon P, Pendem N, Miclet E, Didierjean C, Ennifar E, Guichard G

The canonical helix of urea oligomers at atomic resolution: insights into folding-induced axial organization Article de journal

Dans: Angew Chem Int Ed Engl, vol. 49, no. 6, p. 1067-70, 2010, ISBN: 20039243, (1521-3773 (Electronic) 1433-7851 (Linking) Journal Article Research Support, Non-U.S. Gov't).

Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Freisz S, Bec G, Radi M, Wolff P, Crespan E, Angeli L, Dumas P, Maga G, Botta M, Ennifar E

Crystal structure of HIV-1 reverse transcriptase bound to a non-nucleoside inhibitor with a novel mechanism of action Article de journal

Dans: Angew Chem Int Ed Engl, vol. 49, no. 10, p. 1805-8, 2010, ISBN: 20135654, (1521-3773 (Electronic) 1433-7851 (Linking) Journal Article Research Support, Non-U.S. Gov't).

Liens | BibTeX | Étiquettes: 3-Ring/*chemistry Humans Indoles/*chemistry *Models, Anti-HIV Agents/*chemistry/therapeutic use Crystallography, Biological *Models, DUMAS, ENNIFAR, Molecular Molecular Structure Nitriles/*chemistry Pyridones/*chemistry Pyrimidines/*chemistry Reverse Transcriptase Inhibitors/*chemistry/therapeutic use Vinyl Compounds/*chemistry, Unité ARN, X-Ray HIV Protease Inhibitors/*chemistry/metabolism/pharmacology HIV Reverse Transcriptase/*chemistry/metabolism Heterocyclic Compounds

Sato Y, Ramalanjaona N, Huet T, Potier N, Osz J, Antony P, Peluso-Iltis C, Poussin-Courmontagne P, Ennifar E, Mely Y, Dejaegere A, Moras D, Rochel N

The "Phantom Effect" of the Rexinoid LG100754: structural and functional insights Article de journal

Dans: PLoS One, vol. 5, no. 11, p. e15119, 2010, ISBN: ISBN/1932-6203 (Electronic) 1932-6203 (Linking).

Résumé | Liens | BibTeX | Étiquettes: Animals Binding Sites Binding, Competitive Fluorescence Polarization Humans Ligands Mice Models, DUMAS, ENNIFAR, Molecular Protein Binding Protein Multimerization Protein Structure, Retinoic Acid/*chemistry/genetics/metabolism Recombinant Proteins/chemistry/metabolism Retinoid X Receptors/*chemistry/genetics/metabolism Retinoids/*chemistry/metabolism Scattering, Small Angle Tetrahydronaphthalenes/*chemistry/metabolism Tretinoin/*chemistry/metabolism X-Ray Diffraction, Tertiary Receptor Cross-Talk Receptors, Unité ARN

2009

Burnouf D. Y., Wagner J. E.

Kinetics of deoxy-CTP incorporation opposite a dG-C8-N-2-aminofluorene adduct by a high-fidelity DNA polymerase Article de journal

Dans: J Mol Biol, vol. 386, no. 4, p. 951-61, 2009, (1089-8638 (Electronic) Journal Article Research Support, Non-U.S. Gov't).

Résumé | BibTeX | Étiquettes: Adducts, Bacillus, Catalytic, Cytidine, Deoxyguanosine/*metabolism, DNA, DNA-Directed, Domain, DUMAS, Elements, Fluorenes/*metabolism, Guanine, Kinetics, Oligonucleotides/metabolism, Phosphorothioate, Polymerase/*metabolism, Specificity, stearothermophilus/enzymology, Substrate, Titrimetry, Triphosphate/*metabolism

Wagner J., Etienne H., Fuchs R. P., Cordonnier A., Burnouf D.

Distinct beta-clamp interactions govern the activities of the Y family PolIV DNA polymerase Article de journal

Dans: Mol Microbiol, vol. 74, no. 5, p. 1143-51, 2009, (1365-2958 (Electronic) 0950-382X (Linking) Journal Article).

Résumé | BibTeX | Étiquettes: DUMAS

Wagner J, Etienne H, Fuchs R P, Cordonnier A, Burnouf D

Distinct beta-clamp interactions govern the activities of the Y family PolIV DNA polymerase Article de journal

Dans: Mol Microbiol, vol. 74, no. 5, p. 1143-1151, 2009, ISBN: 19843218, (1365-2958 (Electronic) 0950-382X (Linking) Journal Article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Radi M, Maga G, Alongi M, Angeli L, Samuele A, Zanoli S, Bellucci L, Tafi A, Casaluce G, Giorgi G, Armand-Ugon M, Gonzalez E, Este J A, Baltzinger M, Bec G, Dumas P, Ennifar E, Botta M

Discovery of chiral cyclopropyl dihydro-alkylthio-benzyl-oxopyrimidine (S-DABO) derivatives as potent HIV-1 reverse transcriptase inhibitors with high activity against clinically relevant mutants Article de journal

Dans: J Med Chem, vol. 52, no. 3, p. 840-851, 2009, ISBN: 19140683, (1520-4804 (Electronic) Journal Article Research Support, Non-U.S. Gov't).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

2007

Ali M B, Chaminade F, Kanevsky I, Ennifar E, Josset L, Ficheux D, Darlix J L, Fosse P

Structural requirements for nucleocapsid protein-mediated dimerization of avian leukosis virus RNA Article de journal

Dans: J Mol Biol, vol. 372, no. 4, p. 1082-96, 2007, ISBN: 17706668.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Bernacchi S, Freisz S, Maechling C, Spiess B, Marquet R, Dumas P, Ennifar E

Aminoglycoside binding to the HIV-1 RNA dimerization initiation site: thermodynamics and effect on the kissing-loop to duplex conversion Article de journal

Dans: Nucleic Acids Res, vol. 35, no. 21, p. 7128-39, 2007, ISBN: 17942426, (1362-4962 (Electronic)).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, MARQUET, Unité ARN

Olieric V, Ennifar E, Meents A, Fleurant M, Besnard C, Pattison P, Schiltz M, Schulze-Briese C, Dumas P

Using X-ray absorption spectra to monitor specific radiation damage to anomalously scattering atoms in macromolecular crystallography Article de journal

Dans: Acta Crystallogr D Biol Crystallogr, vol. 63, no. Pt 7, p. 759-68, 2007, ISBN: 17582167.

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Reblova K, Fadrna E, Sarzynska J, Kulinski T, Kulhanek P, Ennifar E, Koca J, Sponer J

Conformations of Flanking Bases in HIV-1 RNA DIS Kissing Complexes Studied by Molecular Dynamics Article de journal

Dans: Biophys J, vol. 93, no. 11, p. 3932-3949, 2007, ISBN: 17704156, (0006-3495 (Print) Journal article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

2006

Ambert N., Vanwinsberghe J., Dumas P.

Biocrystallographica, a package for doing crystallography with Mathematica Divers

2006.

BibTeX | Étiquettes: DUMAS

Dumas P., Vanwinsberghe J., Cura V.

Einstein's tongue for teaching crystallography to biologists Divers

2006.

BibTeX | Étiquettes: DUMAS

Ambert N, Vanwinsberghe J, Dumas P

Biocrystallographica, a package for doing crystallography with Mathematica Divers

2006.

BibTeX | Étiquettes: DUMAS

Dumas P, Vanwinsberghe J, Cura V

Einstein's tongue for teaching crystallography to biologists Divers

2006.

BibTeX | Étiquettes: DUMAS

Ambert N, Vanwinsberghe J, Dumas P

Biocrystallographica, a package for doing crystallography with Mathematica Divers

2006.

BibTeX | Étiquettes: DUMAS

Dumas P, Vanwinsberghe J, Cura V

Einstein's tongue for teaching crystallography to biologists Divers

2006.

BibTeX | Étiquettes: DUMAS

Ennifar E, Dumas P

Polymorphism of bulged-out residues in HIV-1 RNA DIS kissing complex and structure comparison with solution studies Article de journal

Dans: J Mol Biol, vol. 356, no. 3, p. 771-782, 2006, ISBN: 16403527, (0022-2836 (Print) Journal Article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Dumas P, Vanwinsberghe J, Cura V

Einstein's tongue for teaching crystallography to biologists Divers

2006.

BibTeX | Étiquettes: DUMAS, Unité ARN

Ambert N, Vanwinsberghe J, Dumas P

Biocrystallographica, a package for doing crystallography with Mathematica Divers

2006.

BibTeX | Étiquettes: DUMAS, Unité ARN

2005

Ennifar E, Basquin J, Birkenbihl R, Suck D

Purification, crystallization and preliminary X-ray diffraction studies of the archaeal virus resolvase SIRV2 Article de journal

Dans: Acta Crystallogr F Struct Biol Commun, vol. 61, no. Pt 5, p. 507-509, 2005, ISBN: 16511081, (1744-3091 (Electronic) Journal Article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

2004

Burnouf D. Y., Olieric V., Wagner J., Fujii S., Reinbolt J., Fuchs R. P., Dumas P.

Structural and biochemical analysis of sliding clamp/ligand interactions suggest a competition between replicative and translesion DNA polymerases Article de journal

Dans: J Mol Biol, vol. 335, no. 5, p. 1187-97, 2004, (0022-2836 Journal Article).

Résumé | BibTeX | Étiquettes: *Binding, Antigen/metabolism, Bacterial/genetics, beta/*chemistry/genetics/*metabolism, Binding, Cell, coli/*enzymology, Competitive, Crystallization, DNA, DUMAS, Escherichia, Fragments/*metabolism, I/metabolism, III/metabolism, Kinetics, ligands, Models, Molecular, Nuclear, Peptide, Polymerase, Proliferating, Protein, Proteins/chemistry/metabolism, Recombinant, Replication/*genetics, Subunits

Delarue M., Dumas P.

On the use of low-frequency normal modes to enforce collective movements in refining macromolecular structural models Article de journal

Dans: Proc Natl Acad Sci U S A, vol. 101, no. 18, p. 6957-62, 2004, (0027-8424 Journal Article).

Résumé | BibTeX | Étiquettes: *Models, Carrier, coli, Computer, Diffraction, DUMAS, Escherichia, Gov't, Molecular, Non-U.S., Proteins/*chemistry, Proteins/chemistry, Simulation, Support, X-Ray

Schiltz M, Dumas P, Ennifar E, Flensburg C, Paciorek W, Vonrhein C, Bricogne G

Phasing in the presence of severe site-specific radiation damage through dose-dependent modelling of heavy atoms Article de journal

Dans: Acta Crystallogr D Biol Crystallogr, vol. 60, no. Pt 6, p. 1024-1031, 2004, ISBN: 15159561, (0907-4449 Journal Article).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN

Ehresmann C, Ehresmann B, Ennifar E, Dumas P, Garber M, Mathy N, Nikulin A, Portier C, Patel D, Serganov A

Molecular mimicry in translational regulation: the case of ribosomal protein S15. Article de journal

Dans: RNA Biol, vol. 1, no. 1, p. 66-73, 2004, ISBN: 17194931, (Epub 2004 May 5.).

Résumé | Liens | BibTeX | Étiquettes: DUMAS, ENNIFAR, Unité ARN